Roidipedia.Compound reference & reporting
06 AUG 2026
CompoundsCompare Anastrozole vs Exemestane
Comparison

Anastrozole vs Exemestane

A neutral, evidence-rated side-by-side of Anastrozole and Exemestane. Figures are typical reference values, not recommendations.

AnastrozoleExemestane
TypeAncillaryAncillary
Evidence levelWell establishedWell established
Primary classAromatase inhibitorAromatase inhibitor
Half-life~46 hours~24 hours (enzyme suppression outlasts plasma levels)
Typical dose0.25–0.5 mg/wk12.5–25 mg/day
AromatisesNo
HepatotoxicityLow
Documented effects22
Documented side effects13

Anastrozole

A non-steroidal aromatase inhibitor used to control oestradiol on aromatising cycles. Effective and well studied — with over-suppression, not under-dosing, the more common error.

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Exemestane

Steroidal, irreversible ('suicidal') aromatase inhibitor developed for post-menopausal breast cancer. In the PED context it is used to blunt oestrogen conversion from aromatising androgens. Because it is androgenic and does not raise SHBG the way non-steroidal AIs can, it is often favoured, but the recurring error is aggressive dosing that crashes oestradiol and produces joint pain, low libido and adverse lipids.

Full Exemestane page →
Reference information, not medical advice.
Anastrozole vs Exemestane: dosing, effects & side effects compared · Roidipedia